Discovery of Potent and Selective Methylenephosphonic Acid CD73 Inhibitors-Reference-Cited by-同舟云学术

Discovery of Potent and Selective Methylenephosphonic Acid CD73 Inhibitors

Published:2021-01-05 Issue:1 Volume:64 Page:845-860
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sharif Ehesan U.¹^ORCID,Kalisiak Jaroslaw¹,Lawson Kenneth V.¹^ORCID,Miles Dillon H.¹,Newcomb Eric¹,Lindsey Erick A.¹,Rosen Brandon R.¹^ORCID,Debien Laurent P. P.¹,Chen Ada¹,Zhao Xiaoning¹,Young Stephen W.¹,Walker Nigel P.¹,Sträter Norbert²^ORCID,Scaletti Emma R.²,Jin Lixia¹,Xu Guifen¹,Leleti Manmohan R.¹,Powers Jay P.¹

Affiliation:

1. Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States

2. Institute of Bioanalytical Chemistry, Center for Biotechnology and Biomedicine, Leipzig University, Deutscher Platz 5, D-04103 Leipzig, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c01835

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1. Ecto-5’-nucleotidase: Structure function relationships

2. Ectonucleotidases in Tumor Cells and Tumor-Associated Immune Cells: An Overview