Backbone Cyclization Turns a Venom Peptide into a Stable and Equipotent Ligand at Both Muscle and Neuronal Nicotinic Receptors-Reference-Cited by-同舟云学术

Backbone Cyclization Turns a Venom Peptide into a Stable and Equipotent Ligand at Both Muscle and Neuronal Nicotinic Receptors

Published:2020-10-16 Issue:21 Volume:63 Page:12682-12692
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Giribaldi Julien¹,Haufe Yves²,Evans Edward R. J.³,Amar Muriel⁴,Durner Anna²,Schmidt Casey³,Faucherre Adèle⁵,Moha Ou Maati Hamid⁵,Enjalbal Christine¹^ORCID,Molgó Jordi⁴^ORCID,Servent Denis⁴,Wilson David T.³,Daly Norelle L.³^ORCID,Nicke Annette²,Dutertre Sébastien¹^ORCID

Affiliation:

1. Institut des Biomolécules Max Mousseron, Université de Montpellier, CNRS, ENSCM, 34095 Montpellier, France

2. Walther Straub Institute of Pharmacology and Toxicology, Faculty of Medicine, LMU Munich, Nußbaumstraße 26, 80336 Munich, Germany

3. Centre for Molecular Therapeutics, Australian Institute of Tropical Health and Medicine, James Cook University, Cairns, Queensland 4878, Australia

4. Département Médicaments et Technologies pour la Santé (DMTS), Université Paris-Saclay, CEA, SIMoS, ERL CNRS 9004, F-91191 Gif sur Yvette, France

5. Département de Physiologie, Institut de Génomique Fonctionnelle, CNRS/INSERM UMR 5203, Université de Montpellier, 34095 Montpellier, France

Funder

Minist?re de l'Enseignement sup?rieur, de la Recherche et de l'Innovation

Agence Nationale de la Recherche

Deutsche Forschungsgemeinschaft

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c00957

Reference43 articles.

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