Structure–Activity Relationship Studies of Coumarin-like Diacid Derivatives as Human G Protein-Coupled Receptor-35 (hGPR35) Agonists and a Consequent New Design Principle-Reference-Cited by-同舟云学术

Structure–Activity Relationship Studies of Coumarin-like Diacid Derivatives as Human G Protein-Coupled Receptor-35 (hGPR35) Agonists and a Consequent New Design Principle

Published:2021-02-25 Issue:5 Volume:64 Page:2634-2647
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wei Lai¹,Hou Tao¹,Li Jiaqi¹,Zhang Xiuli²,Zhou Han¹,Wang Zhenyu³^ORCID,Cheng Junxiang⁴,Xiang Kaijing¹,Wang Jixia¹,Zhao Yaopeng¹⁴,Liang Xinmiao¹⁴^ORCID

Affiliation:

1. Key Lab of Separation Science for Analytical Chemistry, Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian 116034, China

2. College of Pharmaceutical Science, Soochow University, Suzhou, Jiangsu 215123, China

3. National Engineering Research Center of Seafood, School of Food Science and Technology, Dalian Polytechnic University, Dalian 116034, China

4. Jiangxi Chinese Medicine Science Center of DICP, CAS, Nanchang 330000, China

Funder

Ministry of Science and Technology of the People's Republic of China

Dalian Institute of Chemical Physics

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c01624

Reference34 articles.

1. Orphan GPCR research

2. Impact of GPCR Structures on Drug Discovery

3. Discovery of Three Novel G-Protein-Coupled Receptor Genes

4. Cloning of a G-protein-coupled receptor that shows an activity to transform NIH3T3 cells and is expressed in gastric cancer cells

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