Identification of First-in-Class Inhibitors of Kallikrein-Related Peptidase 6 That Promote Oligodendrocyte Differentiation-Reference-Cited by-同舟云学术

Identification of First-in-Class Inhibitors of Kallikrein-Related Peptidase 6 That Promote Oligodendrocyte Differentiation

Published:2021-05-05 Issue:9 Volume:64 Page:5667-5688
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Aït Amiri Sabrina¹,Deboux Cyrille²,Soualmia Feryel¹,Chaaya Nancy¹,Louet Maxime³,Duplus Eric¹,Betuing Sandrine⁴,Nait Oumesmar Brahim²,Masurier Nicolas³,El Amri Chahrazade¹^ORCID

Affiliation:

1. Faculty of Sciences and Engineering, IBPS, UMR 8256 CNRS-UPMC, ERL INSERM U1164, Biological Adaptation and Ageing, Sorbonne Université, F-75252 Paris, France

2. Institut du Cerveau, Inserm U 1127, CNRS UMR 7725, Sorbonne Université, F-75013 Paris, France

3. Institut des Biomolécules Max Mousseron, Université de Montpellier, CNRS, ENSCM, F-34093 Montpellier, France

4. Faculty of Sciences and Engineering, IBPS, UMR 8246-CNRS/INSERM U1130, Neurosciences Paris Seine, Sorbonne Université, F-75252 Paris, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c02175

Reference53 articles.

1. Multiple Sclerosis Pathology

2. Mechanisms of neurodegeneration and axonal dysfunction in multiple sclerosis

3. Differentiation block of oligodendroglial progenitor cells as a cause for remyelination failure in chronic multiple sclerosis

4. Remyelinating Pharmacotherapies in Multiple Sclerosis

5. Drug discovery for remyelination and treatment of MS

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