An in Vitro and in Vivo Investigation of Bivalent Ligands That Display Preferential Binding and Functional Activity for Different Melanocortin Receptor Homodimers-Reference-Cited by-同舟云学术

An in Vitro and in Vivo Investigation of Bivalent Ligands That Display Preferential Binding and Functional Activity for Different Melanocortin Receptor Homodimers

Published:2016-03-29 Issue:7 Volume:59 Page:3112-3128
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Lensing Cody J.¹,Freeman Katie T.¹,Schnell Sathya M.¹,Adank Danielle N.¹,Speth Robert C.²³,Haskell-Luevano Carrie¹

Affiliation:

1. Department of Medicinal Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States

2. College of Pharmacy, Nova Southeastern University, Fort Lauderdale, Florida 33328-2018, United States

3. Department of Pharmacology and Physiology, Georgetown University, Washington, D.C. 20057, United States

Funder

National Institute of Diabetes and Digestive and Kidney Diseases

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b01894

Reference110 articles.

1. The Cloning of a Family of Genes That Encode the Melanocortin Receptors

2. Effect of Alpha- and Beta-Melanocyte Stimulating Hormones on the Skin Colour of Man

3. A role for the melanocortin 4 receptor in sexual function

4. Modulation of Blood Pressure by Central Melanocortinergic Pathways

5. Memory impairment induced by IL-1β is reversed by α-MSH through central melanocortin-4 receptors

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