Evaluation of 3-Ethyl-3-(phenylpiperazinylbutyl)oxindoles as PET Ligands for the Serotonin 5-HT7 Receptor: Synthesis, Pharmacology, Radiolabeling, and in Vivo Brain Imaging in Pigs

Author:

Herth Matthias M.12,Andersen Valdemar L.12,Hansen Hanne D.1,Stroth Nikolas3,Volk Balázs4,Lehel Szabolcs5,Dyssegaard Agnete1,Ettrup Anders1,Svenningsson Per3,Knudsen Gitte M.1,Kristensen Jesper L.12

Affiliation:

1. Center for Integrated Molecular Brain Imaging, Rigshospitalet and University of Copenhagen, Blegdamsvej 9, DK-2100 Copenhagen, Denmark

2. Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Universitetsparken 2, DK-2100 Copenhagen, Denmark

3. Center for Molecular Medicine, Department of Neurology and Clinical Neuroscience, Karolinska Institute and Karolinska University Hospital, 17176 Stockholm, Sweden

4. Egis Pharmaceuticals Plc, P.O. Box 100, H-1475 Budapest, Hungary

5. PET and Cyclotron Unit, Rigshospitalet, Blegdamsvej 9, DK-2100 Copenhagen, Denmark

Funder

European Commission Directorate-General for Research and Innovation

Lundbeckfonden

Det Sundhedsvidenskabelige Fakultet, Københavns Universitet

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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