Mimicking of Arginine by Functionalized Nω-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples-Reference-Cited by-同舟云学术

Mimicking of Arginine by Functionalized Nω-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples

Published:2016-02-11 Issue:5 Volume:59 Page:1925-1945
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Keller Max¹,Kuhn Kilian K.¹,Einsiedel Jürgen²,Hübner Harald²,Biselli Sabrina¹,Mollereau Catherine³,Wifling David¹,Svobodová Jaroslava¹,Bernhardt Günther¹,Cabrele Chiara⁴,Vanderheyden Patrick M. L.⁵,Gmeiner Peter²,Buschauer Armin¹

Affiliation:

1. Institute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Universitätsstrasse 31, D-93053 Regensburg, Germany

2. Department of Chemistry and Pharmacy, Emil Fischer Center, Friedrich Alexander University, Schuhstrasse 19, D-91052 Erlangen, Germany

3. Institut de Pharmacologie et Biologie Structurale, CNRS/IPBS, 205 route de Narbonne, 31077 Toulouse cedex 5, France

4. Department of Molecular Biology, University of Salzburg, Billrothstrasse 11, A-5020 Salzburg, Austria

5. Faculty of Sciences and Bioengineering Sciences, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium

Funder

Deutsche Forschungsgemeinschaft

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b01495

Reference86 articles.

1. The Bolton and Hunter Method for Radiolabeling Protein

2. Differential Conjugation of Tat Peptide to Superparamagnetic Nanoparticles and Its Effect on Cellular Uptake

3. Novel modified and radiolabelled neuropeptide Y analogues to study Y-receptor subtypes

4. A Simple and Powerful Flow Cytometric Method for the Simultaneous Determination of Multiple Parameters at G Protein-Coupled Receptor Subtypes

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