Improving the Selectivity of Engineered Protease Inhibitors: Optimizing the P2 Prime Residue Using a Versatile Cyclic Peptide Library-Reference-Cited by-同舟云学术

Improving the Selectivity of Engineered Protease Inhibitors: Optimizing the P2 Prime Residue Using a Versatile Cyclic Peptide Library

Published:2015-10-05 Issue:20 Volume:58 Page:8257-8268
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

de Veer Simon J.¹,Wang Conan K.²,Harris Jonathan M.¹,Craik David J.²,Swedberg Joakim E.²

Affiliation:

1. Institute of Health and Biomedical Innovation, Queensland University of Technology, Brisbane, Queensland QLD 4059, Australia

2. Institute for Molecular Bioscience, The University of Queensland, 306 Carmody Road, Building 80, Queensland Bioscience Presinct, Brisbane, Queensland, QLD 4072, Australia

Funder

National Health and Medical Research Council

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b01148

Reference62 articles.

1. The pharmacological landscape and therapeutic potential of serine hydrolases

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