Fragment-Based Discovery of 2-Aminoquinazolin-4(3H)-ones As Novel Class Nonpeptidomimetic Inhibitors of the Plasmepsins I, II, and IV-Reference-Cited by-同舟云学术

Fragment-Based Discovery of 2-Aminoquinazolin-4(3H)-ones As Novel Class Nonpeptidomimetic Inhibitors of the Plasmepsins I, II, and IV

Published:2015-12-23 Issue:1 Volume:59 Page:374-387
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rasina Dace¹,Otikovs Martins¹,Leitans Janis²,Recacha Rosario¹,Borysov Oleksandr V.¹,Kanepe-Lapsa Iveta¹,Domraceva Ilona¹,Pantelejevs Teodors¹,Tars Kaspars²,Blackman Michael J.³,Jaudzems Kristaps¹,Jirgensons Aigars¹

Affiliation:

1. Latvian Institute of Organic Synthesis, Aizkraukles 21, Riga LV-1006, Latvia

2. Biomedical Research and Study Centre, Ratsupites 1, Riga LV-1067, Latvia

3. The Francis Crick Institute, Mill Hill Laboratory, The Ridgeway, Mill Hill, London NW7 1AA, U.K.

Funder

European Regional Development Fund

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b01558

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