Chiral Dihydrobenzofuran Acids Show Potent Retinoid X Receptor–Nuclear Receptor Related 1 Protein Dimer Activation

Author:

Sundén Henrik1,Schäfer Anja12,Scheepstra Marcel2,Leysen Seppe2,Malo Marcus1,Ma Jian-Nong3,Burstein Ethan S.3,Ottmann Christian2,Brunsveld Luc2,Olsson Roger134

Affiliation:

1. Department of Chemistry and Molecular Biology, Medicinal Chemistry, University of Gothenburg, SE-41296 Gothenburg, Sweden

2. Department of Biomedical Engineering and Institute of Complex Molecular Systems, Laboratory of Chemical Biology, Technische Universiteit Eindhoven, Den Dolech 2, 5612 AZ Eindhoven, The Netherlands

3. ACADIA Pharmaceuticals Inc., San Diego, California 92130, United States

4. Chemical Biology & Therapeutics, Department of Experimental Medical Science, Lund University, Sölvegatan 19, BMC DIO, SE-221 84 Lund, Sweden

Funder

Vetenskapsr?det

Michael J. Fox Foundation for Parkinson's Research

Directorate-General for Research and Innovation

Nederlandse Organisatie voor Wetenschappelijk Onderzoek

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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