Discovery and Characterization of Biased Allosteric Agonists of the Chemokine Receptor CXCR3

Author:

Milanos Lampros1,Brox Regine1,Frank Theresa1,Poklukar Gašper12,Palmisano Ralf3,Waibel Reiner1,Einsiedel Jürgen1,Dürr Maximilian4,Ivanović-Burmazović Ivana4,Larsen Olav5,Hjortø Gertrud Malene5,Rosenkilde Mette Marie5,Tschammer Nuska1

Affiliation:

1. Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University, Schuhstraße 19, 91052 Erlangen, Germany

2. Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia

3. Optical Imaging Center Erlangen, Friedrich Alexander University, Hartmannstraße 14, 91052 Erlangen, Germany

4. Department of Chemistry and Pharmacy, Bioorganic Chemistry, Friedrich Alexander University, Egerlandstraße 1, 91058 Erlangen, Germany

5. Department of Neuroscience and Pharmacology, Laboratory for Molecular Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Blegdamsvej 3B, DK-2200 Copenhagen N, Denmark

Funder

Deutsche Forschungsgemeinschaft

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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