Development of Fluorescent 4-[4-(3<i>H</i>-Spiro[isobenzofuran-1,4′-piperidin]-1′-yl)butyl]indolyl Derivatives as High-Affinity Probes to Enable the Study of σ Receptors via Fluorescence-Based Techniques-Reference-Cited by-同舟云学术

Development of Fluorescent 4-[4-(3H-Spiro[isobenzofuran-1,4′-piperidin]-1′-yl)butyl]indolyl Derivatives as High-Affinity Probes to Enable the Study of σ Receptors via Fluorescence-Based Techniques

Published:2023-03-15 Issue:6 Volume:66 Page:3798-3817
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Abatematteo Francesca Serena¹,Majellaro Maria²,Montsch Bianca³,Prieto-Díaz Rubén²^ORCID,Niso Mauro¹,Contino Marialessandra¹^ORCID,Stefanachi Angela¹^ORCID,Riganti Chiara⁴^ORCID,Mangiatordi Giuseppe Felice⁵^ORCID,Delre Pietro⁵,Heffeter Petra³,Sotelo Eddy²^ORCID,Abate Carmen¹⁵^ORCID

Affiliation:

1. Dipartimento di Farmacia-Scienze del Farmaco, Via Orabona, 4, 79125 Bari, Italy

2. Centro Singular Investigación Quimica Biologica e Materiales Moleculares (CIQUS), Departamento de Quimica Orgánica, Facultade de Farmacia, Universidade de Santiago de Compostela, 15782 Santiago de Compostela, Spain

3. Center for Cancer Research and Comprehensive Cancer Center, Medical University of Vienna, Borschkegasse 8a, 1090 Vienna, Austria

4. Department of Oncology, University of Torino, via Santena 5/bis, 10126 Torino, Italy

5. Consiglio Nazionale delle Ricerche (CNR), Istituto di Cristallografia, Via Amendola, 70126 Bari, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c01227

Reference75 articles.

1. Editorial [Hot topic: Sigma1 and Sigma 2 Receptors (Guest Editor: Richard A. Glennon)]

2. Purification, molecular cloning, and expression of the mammalian sigma1-binding site.

3. Crystal structure of the human σ1 receptor

4. The Molecular Function of σ Receptors: Past, Present, and Future

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