[1,2,4]Triazolo[3,4-<i>b</i>]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes-Reference-Cited by-同舟云学术

[1,2,4]Triazolo[3,4-b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes

Published:2023-01-04 Issue:2 Volume:66 Page:1301-1320
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Murthy Sudarshan¹,Nizi Maria Giulia²,Maksimainen Mirko M.¹,Massari Serena²^ORCID,Alaviuhkola Juho¹,Lippok Barbara E.³,Vagaggini Chiara⁴,Sowa Sven T.¹,Galera-Prat Albert¹,Ashok Yashwanth¹^ORCID,Venkannagari Harikanth¹^ORCID,Prunskaite-Hyyryläinen Renata¹,Dreassi Elena⁴,Lüscher Bernhard³^ORCID,Korn Patricia³,Tabarrini Oriana²^ORCID,Lehtiö Lari¹^ORCID

Affiliation:

1. Faculty of Biochemistry and Molecular Medicine and Biocenter Oulu, University of Oulu, Oulu90220, Finland

2. Department of Pharmaceutical Sciences, University of Perugia, Perugia06123, Italy

3. Institute of Biochemistry and Molecular Biology, RWTH Aachen University, Aachen52074, Germany

4. Department of Biotechnology, Chemistry and Pharmacy, University of Siena, SienaI-53100, Italy

Funder

Sigrid Jus?liuksen S??ti?

Deutsche Forschungsgemeinschaft

Jane ja Aatos Erkon S??ti?

Magnus Ehrnroothin S??ti?

Publisher

American Chemical Society (ACS)