Discovery of Highly Selective Inhibitors of the Human Constitutive Proteasome β5c Chymotryptic Subunit-Reference-Cited by-同舟云学术

Discovery of Highly Selective Inhibitors of the Human Constitutive Proteasome β5c Chymotryptic Subunit

Published:2023-01-06 Issue:2 Volume:66 Page:1172-1185
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zhan Wenhu¹^ORCID,Li Daqiang¹^ORCID,Saha Priya¹,Wang Rong²,Zhang Hao¹^ORCID,Ajay Amrendra K.³^ORCID,Deban Christa⁴,Sukenick George²,Azzi Jamil³,Lin Gang¹^ORCID

Affiliation:

1. Department of Microbiology & Immunology, Weill Cornell Medicine, 1300 York Ave., New York, New York 10065, United States

2. NMR Analytical Core Facility, Memorial Sloan Kettering Cancer Center, New York, New York 10065, United States

3. Renal Division, Brigham and Women’s Hospital, Harvard Medical School, Boston, Massachusetts 02115, United States

4. Transplantation Research Center, Renal Division, Brigham and Women’s Hospital, Harvard Medical School, Boston, Massachusetts 02115, United States

Funder

National Cancer Institute

National Institute of Allergy and Infectious Diseases

Talal and Maha Shair foundation

The Daedalus Fund for Innovation of Weill Cornell Medicine

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c00733

Reference42 articles.

1. The Proteasome: Paradigm of a Self-Compartmentalizing Protease

2. The unique functions of tissue-specific proteasomes

3. Proteasomes in immune cells: more than peptide producers?

4. Regulation of CD8 + T Cell Development by Thymus-Specific Proteasomes

5. Acetylation-Mediated Proteasomal Degradation of Core Histones during DNA Repair and Spermatogenesis

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