Highly Potent and Selective Dopamine D4 Receptor Antagonists Potentially Useful for the Treatment of Glioblastoma

Author:

Pavletić Pegi1,Semeano Ana2,Yano Hideaki2,Bonifazi Alessandro3ORCID,Giorgioni Gianfabio1ORCID,Piergentili Alessandro1ORCID,Quaglia Wilma1ORCID,Sabbieti Maria Giovanna4,Agas Dimitrios4,Santoni Giorgio1,Pallini Roberto56,Ricci-Vitiani Lucia7,Sabato Emanuela8,Vistoli Giulio8ORCID,Del Bello Fabio1ORCID

Affiliation:

1. Scuola di Scienze del Farmaco e dei Prodotti della Salute, Università di Camerino,, Camerino 62032, Italy

2. Department of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, Bouvé College of Health Sciences, Center for Drug Discovery, Northeastern University, Boston, Massachusetts 02115, United States

3. Medicinal Chemistry Section, Molecular Targets and Medications Discovery Branch, National Institute on Drug Abuse−Intramural Research Program, National Institutes of Health, 333 Cassell Drive, Baltimore, Maryland 21224, United States

4. Scuola di Bioscienze e Medicina Veterinaria, Università di Camerino, Via Gentile III da Varano, Camerino 62032, Italy

5. Institute of Neurosurgery, Scientific Hospitalization and Care Institute (IRCCS), Gemelli University Polyclinic Foundation, Rome 00168, Italy

6. Institute of Neurosurgery, School of Medicine, Catholic University, Rome 00168, Italy

7. Department of Hematology, Oncology and Molecular Medicine, Istituto Superiore di Sanità, Rome 00161, Italy

8. Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Mangiagalli 25, Milano 20133, Italy

Funder

Universit? degli Studi di Camerino

National Institute on Drug Abuse

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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