Metabolism-Guided Selective Androgen Receptor Antagonists: Design, Synthesis, and Biological Evaluation for Activity against Enzalutamide-Resistant Prostate Cancer-Reference-Cited by-同舟云学术

Metabolism-Guided Selective Androgen Receptor Antagonists: Design, Synthesis, and Biological Evaluation for Activity against Enzalutamide-Resistant Prostate Cancer

Published:2023-02-24 Issue:5 Volume:66 Page:3372-3392
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hwang Dong-Jin¹^ORCID,He Yali¹,Ponnusamy Suriyan²,Thiyagarajan Thirumagal²,Mohler Michael L.¹^ORCID,Narayanan Ramesh²,Miller Duane D.¹^ORCID

Affiliation:

1. Department of Pharmaceutical Sciences, University of Tennessee Health Science Center, Memphis, Tennessee 38163, United States

2. Department of Medicine, University of Tennessee Health Science Center, Memphis, Tennessee 38163, United States

Funder

National Cancer Institute

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c01858

Reference37 articles.

1. Eighty Years of Targeting Androgen Receptor Activity in Prostate Cancer: The Fight Goes on

2. Cancer treatment and survivorship statistics, 2019

3. Androgen receptor: A key molecule in the progression of prostate cancer to hormone independence

4. Role of Androgen Receptor in Prostate Cancer: A Review

5. Bicalutamide

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