Identification of TUL01101: A Novel Potent and Selective JAK1 Inhibitor for the Treatment of Rheumatoid Arthritis-Reference-Cited by-同舟云学术

Identification of TUL01101: A Novel Potent and Selective JAK1 Inhibitor for the Treatment of Rheumatoid Arthritis

Published:2022-12-13 Issue:24 Volume:65 Page:16716-16740
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zhou Shuhao¹,Mao Weiwei²,Su Yuan¹,Zheng Xuejian²,Qian Wenyuan²,Shen Meiyue¹,Shan Ningli¹,Li Yaoshuang¹,Wang Degang¹,Wu Shouting¹,Sun Tiemin³^ORCID,Mu Liwei¹^ORCID

Affiliation:

1. Zhuhai United Laboratories Co., Ltd., NO.12 Jialian Road, Tanzhou Township, Zhongshan, Guangdong 528467, P. R. China

2. WuXi AppTec (Shanghai) Co., Ltd., 288 FuTe Zhong Road, Shanghai 200131, P. R. China

3. Key Laboratory of Structure-Based Drug Design and Discovery, Shenyang Pharmaceutical University, Ministry of Education, Shenyang 110016, P. R. China

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c01550

Reference50 articles.

1. Rheumatoid arthritis pathophysiology: update on emerging cytokine and cytokine-associated cell targets

2. The Pathogenesis of Rheumatoid Arthritis

3. Synthesis and Evaluation of Hydrogen Peroxide Sensitive Prodrugs of Methotrexate and Aminopterin for the Treatment of Rheumatoid Arthritis

4. The comparative effectiveness of abatacept versus anti-tumour necrosis factor switching for rheumatoid arthritis patients previously treated with an anti-tumour necrosis factor

5. Biologic Rheumatoid Arthritis Therapies

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