Novel Antagonist of the Type 2 Lysophosphatidic Acid Receptor (LPA2), UCM-14216, Ameliorates Spinal Cord Injury in Mice

Author:

Khiar-Fernández Nora1,Zian Debora1,Vázquez-Villa Henar1ORCID,Martínez R. Fernando1ORCID,Escobar-Peña Andrea1,Foronda-Sainz Román1,Ray Manisha2,Puigdomenech-Poch Maria3,Cincilla Giovanni4ORCID,Sánchez-Martínez Melchor45ORCID,Kihara Yasuyuki2,Chun Jerold2,López-Vales Rubèn3ORCID,López-Rodríguez María L.1ORCID,Ortega-Gutiérrez Silvia1ORCID

Affiliation:

1. Departamento de Química Orgánica I, Facultad de Ciencias Químicas, Universidad Complutense de Madrid, Madrid E-28040, Spain

2. Translational Neuroscience Initiative, Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States

3. Departament de Biologia Cel·lular, Fisiologia i Immunologia, Institut de Neurociències, Centro de Investigación Biomédica en Red sobre Enfermedades Neurodegenerativas (CIBERNED), Universitat Autònoma de Barcelona, Bellaterra, BarcelonaE-08193, Spain

4. Molomics, Barcelona Science Park, Baldiri i Reixac 4-8, Barcelona E-08028, Spain

5. Burua Scientific, Sant Pere de Ribes E-08810, Spain

Funder

National Institute of Neurological Disorders and Stroke

Comunidad de Madrid

U.S. Department of Defense

National Institute of Mental Health

Instituci? Catalana de Recerca i Estudis Avan?ats

Agencia Estatal de Investigaci?n,Ministerio de Ciencia, Innovaci?n y Universidades

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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