Design, Synthesis, Biological Activity, and Structural Analysis of Novel Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D<sub>3</sub>-Reference-Cited by-同舟云学术

Design, Synthesis, Biological Activity, and Structural Analysis of Novel Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D₃

Published:2022-09-27 Issue:19 Volume:65 Page:13112-13124
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Seoane Samuel¹,Gogoi Pranjal²,Zárate-Ruíz Araceli²,Peluso-Iltis Carole³,Peters Stefan²^ORCID,Guiberteau Thierry⁴,Maestro Miguel A.⁵,Pérez-Fernández Román¹,Rochel Natacha³^ORCID,Mouriño Antonio²

Affiliation:

1. Department of Physiology−Center for Research in Molecular Medicine and Chronic Diseases (CIMUS), University of Santiago de Compostela, Avda. Barcelona s/n, Santiago de Compostela 15706, Spain

2. Department of Organic Chemistry, Research Laboratory Ignacio Ribas, University of Santiago de Compostela, Avda. de las Ciencias s/n, Santiago de Compostela 15782, Spain

3. Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC); Institut National de La Santé et de La Recherche Médicale (INSERM), U1258; Centre National de Recherche Scientifique (CNRS), UMR7104, Université de Strasbourg, Strasbourg, Illkirch 67400, France

4. Laboratoire ICube─Université de Strasbourg, CNRS UMR 7357, Strasbourg 67000, France

5. Department of Chemistry-CICA, University of A Coruña, Campus da Zapateira s/n, A Coruña 15071, Spain

Funder

Agence Nationale de la Recherche

Deutscher Akademischer Austauschdienst

Agencia Estatal de Investigaci?n

European Regional Development Fund

Xunta de Galicia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c00900

Reference79 articles.

1. The History of the Discovery of Vitamin D and Its Daughter Steroid Hormone

2. Sunlight and Vitamin D

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4. The discovery and synthesis of the nutritional factor vitamin D

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