Two Decades of Successful SAR-Grounded Stories of the Novel Bacterial Topoisomerase Inhibitors (NBTIs)-Reference-Cited by-同舟云学术

Two Decades of Successful SAR-Grounded Stories of the Novel Bacterial Topoisomerase Inhibitors (NBTIs)

Published:2020-02-06 Issue:11 Volume:63 Page:5664-5674
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Kolarič Anja¹²,Anderluh Marko²^ORCID,Minovski Nikola¹^ORCID

Affiliation:

1. Laboratory for Cheminformatics, Theory Department, National Institute of Chemistry, Hajdrihova 19, SI-1001 Ljubljana, Slovenia

2. Chair of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, SI-1000 Ljubljana, Slovenia

Funder

Javna Agencija za Raziskovalno Dejavnost RS

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b01738

Reference52 articles.

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3. Malleron, J.L.; Tabart, M.; Carry, J. C.; Evers, M.; El Ahmad, Y.; Mignani, S.; Viviani, F. Quinolyl Propyl Piperidine Derivatives And Theiruse As Antibacterial Agents. Patent WO 200125227, 2001.

4. Type IIA topoisomerase inhibition by a new class of antibacterial agents

5. Design, Synthesis, and Characterization of Novel Tetrahydropyran-Based Bacterial Topoisomerase Inhibitors with Potent Anti-Gram-Positive Activity

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