Kinase Atlas: Druggability Analysis of Potential Allosteric Sites in Kinases

Author:

Yueh Christine,Rettenmaier Justin1,Xia Bing,Hall David R.2,Alekseenko Andrey,Porter Kathryn A.,Barkovich Krister1,Keseru Gyorgy3,Whitty AdrianORCID,Wells James A.1,Vajda SandorORCID,Kozakov DimaORCID

Affiliation:

1. Departments of Pharmaceutical Chemistry and Cellular and Molecular Pharmacology, University of California, 1700 Fourth Street, San Francisco, California 9415, United States

2. Acpharis Incorporated, Holliston, Massachusetts 01746, United States

3. Medicinal Chemistry Research Group, Research Center for Natural Sciences, Magyar tudósok krt. 2, H-1117 Budapest, Hungary

Funder

Division of Computing and Communication Foundations

National Institute of General Medical Sciences

National Research, Development and Innovation Office of Hungary

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Reference69 articles.

1. Classification of small molecule protein kinase inhibitors based upon the structures of their drug-enzyme complexes

2. Human Protein Kinase Knowledgebase. http://www.kinasenet.ca (accessed May 13, 2019).

3. The Protein Kinase Complement of the Human Genome

4. Comprehensive Structural and Functional Characterization of the Human Kinome by Protein Structure Modeling and Ligand Virtual Screening

5. Blue Ridge Institute for Medical Research. FDA-approved protein kinase inhibitors. http://www.brimr.org/PKI/PKIs.htm (accessed May 13, 2019).

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