Structure-Based Optimization of Coumarin hA3 Adenosine Receptor Antagonists-Reference-Cited by-同舟云学术

Structure-Based Optimization of Coumarin hA3 Adenosine Receptor Antagonists

Published:2019-11-18 Issue:5 Volume:63 Page:2577-2587
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Matos Maria João¹²^ORCID,Vilar Santiago²,Vazquez-Rodriguez Saleta²,Kachler Sonja³,Klotz Karl-Norbert³^ORCID,Buccioni Michela⁴,Delogu Giovanna⁵^ORCID,Santana Lourdes²,Uriarte Eugenio²⁶,Borges Fernanda¹^ORCID

Affiliation:

1. CIQUP/Department of Chemistry and Biochemistry, Faculty of Sciences, University of Porto, 4169-007 Porto, Portugal

2. Department of Organic Chemistry, Faculty of Pharmacy, University of Santiago de Compostela, 15782 Santiago de Compostela, Spain

3. Institute of Pharmacology and Toxicology, University of Würzburg, 97078 Würzburg, Germany

4. School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, 62032 Camerino, Italy

5. Department of Life Sciences and Environment—Section of Pharmaceutical Sciences, University of Cagliari, 09124 Cagliari, Italy

6. Instituto de Ciencias Químicas Aplicadas, Universidad Autónoma de Chile, 7500912 Santiago, Chile

Funder

European Regional Development Fund

H2020 Marie Sklodowska-Curie Actions

Universidade do Porto

European Social Fund

Funda??o para a Ci?ncia e a Tecnologia

Conseller?a de Cultura, Educaci?n e Ordenaci?n Universitaria, Xunta de Galicia

University of Santiago de Compostela

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b01572

Reference50 articles.

1. Adenosine Receptors: Expression, Function and Regulation

2. International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors—An Update

3. Functionally biased modulation of A3 adenosine receptor agonist efficacy and potency by imidazoquinolinamine allosteric enhancers

4. Adenosine receptors as drug targets — what are the challenges?

5. Mechanisms of induction of adenosine receptor genes and its functional significance

Cited by 16 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Benzopyrone, a privileged scaffold in drug discovery: An overview of FDA‐approved drugs and clinical candidates;Medicinal Research Reviews;2024-03-26

2. Exploring Urease Inhibition by Coumarin Derivatives through in silico and in vitro Methods;Journal of the Brazilian Chemical Society;2024

3. Evaluation of in vitro cytotoxic and genotoxic effects of the 3‐(3,4‐dihydroxyphenyl)‐8‐hydroxycoumarin;Journal of Applied Toxicology;2023-05-08

4. Cytogenotoxicity assessment of 3‐(3,4‐dihydroxyphenyl)‐7,8‐dihydroxycoumarin on HepG2/C3A cells and leukocytes;Journal of Applied Toxicology;2022-09-02

5. Deep-red/NIR emitting coumarin derivatives - Synthesis, photophysical properties, and biological applications;Dyes and Pigments;2022-06