Identification and Optimization of Novel Cathepsin C Inhibitors Derived from EGFR Inhibitors
Author:
Affiliation:
1. National Institute of Biological Sciences (NIBS), 7 Science Park Road, ZGC Life Science Park, Beijing 102206, China
Funder
Ministry of Science and Technology of the People's Republic of China
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b00631
Reference36 articles.
1. Structure of human dipeptidyl peptidase I (cathepsin C): exclusion domain added to an endopeptidase framework creates the machine for activation of granular serine proteases
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