Design, Synthesis, and Optimization of Balanced Dual NK1/NK3 Receptor Antagonists-Reference-Cited by-同舟云学术

Design, Synthesis, and Optimization of Balanced Dual NK1/NK3 Receptor Antagonists

Published:2014-02-13 Issue:5 Volume:5 Page:550-555
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Hanessian Stephen¹,Jennequin Thomas¹,Boyer Nicolas¹,Babonneau Vincent¹,Soma Udaykumar¹,Mannoury la Cour Clotilde²,Millan Mark J.²,De Nanteuil Guillaume³

Affiliation:

1. Department of Chemistry, Université de Montréal, Station Centre-Ville, Montréal, Que. H3C 3J7, Canada

2. Department of Psychopharmacology, Institut de Recherches Servier, 125 Chemin de Ronde, 78290 Croissy-sur-Seine, France

3. Neuroscience Chemistry Research Unit, Institut de Recherches Servier, 125 Chemin de Ronde, 78290 Croissy-sur-Seine, France

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml400528y

Reference60 articles.

1. Tachykinins and Tachykinin Receptors: Structure and Activity Relationships

2. The NK1 receptor antagonist WIN51708 reduces sensitization after chronic cocaine

3. NK3 receptor antagonists: the next generation of antipsychotics?

4. Therapeutic Utility of NK3 Receptor Antagonists for the Treatment of Schizophrenia

5. For an example of dual NK1/NK3 antagonists for the treatment of Schizophrenia, see also:Alvaro, G.; Andreotti, A.; Belvedere, S.; Di Fabio, R.; Falchi, A.; Giovannini, R.Pyridine derivatives and their use in the treatment of psychotic disorders. WO2007028654, 2007.

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