Synthesis and Biological Evaluation of the Enantiomers of the Potent and Selective A1-Adenosine Antagonist 1,3-Dipropyl-8-[2-(5,6-epoxynorbonyl)]- xanthine-Reference-Cited by-同舟云学术

Synthesis and Biological Evaluation of the Enantiomers of the Potent and Selective A1-Adenosine Antagonist 1,3-Dipropyl-8-[2-(5,6-epoxynorbonyl)]- xanthine

Published:1997-06-01 Issue:12 Volume:40 Page:1773-1778
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Pfister Jürg R.¹,Belardinelli Luiz¹,Lee Gavin¹,Lum Robert T.¹,Milner Peter¹,Stanley William C.¹,Linden Joel¹,Baker Stephen P.¹,Schreiner George¹

Affiliation:

1. CV Therapeutics, Palo Alto, California 94304, Departments of Medicine and Pharmacology, College of Medicine, University of Florida, Gainesville, Florida 32610, and University of Virginia School of Medicine, Charlottesville, Virginia 22908

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970013w

Reference37 articles.

1. Inhibitors of gastric acid secretion: 3,4-diamino-1,2,5-thiadiazole 1-oxides and 1,1-dioxides as urea equivalents in a series of histamine H2 receptor antagonists

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