Improved Synthesis of N-Benzylaminoferrocene-Based Prodrugs and Evaluation of Their Toxicity and Antileukemic Activity

Author:

Daum Steffen1,Chekhun Vasiliy F.2,Todor Igor N.2,Lukianova Natalia Yu.2,Shvets Yulia V.2,Sellner Leopold34,Putzker Kerstin5,Lewis Joe5,Zenz Thorsten34,de Graaf Inge A. M.6,Groothuis Geny M. M.6,Casini Angela6,Zozulia Oleksii1,Hampel Frank1,Mokhir Andriy1

Affiliation:

1. Department of Chemistry and Pharmacy, Organic Chemistry II, Friedrich-Alexander-University of Erlangen-Nürnberg, Henkestraße 42, 91054 Erlangen, Germany

2. R. E. Kavetsky Institute of Experimental Pathology, Oncology, and Radiobiology of the National Academy of Sciences of Ukraine, Vasilkivska 45, 03022 Kyiv, Ukraine

3. Department of Translational Oncology, National Center for Tumor Diseases (NCT) and German Cancer Research Center (DKFZ) Heidelberg, Im Neuenheimer Feld 460, 69120 Heidelberg, Germany

4. Department of Medicine V, University Hospital Heidelberg, Im Neuenheimer Feld 410, 69120 Heidelberg, Germany

5. Chemical Biology Core Facility, European Molecular Biology Laboratory Heidelberg, Meyerhofstraße 1, 69117 Heidelberg, Germany

6. Department of Pharmacokinetics, Toxicology and Targeting, Groningen Research Institute of Pharmacy, University of Groningen, A. Deusinglaan 1, 9713 AV Groningen, The Netherlands

Funder

European Commission

European Cooperation in Science and Technology

Friedrich-Alexander-Universität Erlangen-Nürnberg

Helmholtz Association

Deutsche Forschungsgemeinschaft

University of Groningen

Dr. Hertha und Helmut Schmauser-Stiftung

Chemical Biology Core Facility

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3