Identification of a Potent and Selective 5-HT1A Receptor Agonist with In Vitro and In Vivo Antinociceptive Activity

Author:

Linciano Pasquale1ORCID,Sorbi Claudia1ORCID,Comitato Antonella2,Lesniak Anna3,Bujalska-Zadrożny Magdalena3,Pawłowska Agata3,Bielenica Anna4,Orzelska-Górka Jolanta5,Kędzierska Ewa5,Biała Grażyna5,Ronsisvalle Simone6ORCID,Limoncella Silvia7,Casarini Livio78,Cichero Elena9,Fossa Paola9,Satała Grzegorz10,Bojarski Andrzej J.10ORCID,Brasili Livio1ORCID,Bardoni Rita2,Franchini Silvia1ORCID

Affiliation:

1. Department of Life Sciences, University of Modena and Reggio Emilia, Via Campi 103, 41125 Modena, Italy

2. Department of Biomedical, Metabolic and Neural Sciences, University of Modena and Reggio Emilia, Via Campi 287, 41125 Modena, Italy

3. Department of Pharmacodynamics, Faculty of Pharmacy, Centre for Preclinical Research and Technology, Medical University of Warsaw, Banacha 1, 02-097 Warsaw, Poland

4. Department of Biochemistry, Medical University of Warsaw, Banacha 1, 02-097 Warsaw, Poland

5. Department of Pharmacology and Pharmacodynamics, Faculty of Pharmacy with Division of Medical Analytics, Medical University of Lublin, Chodzki 4A, 20-093 Lublin, Poland

6. Department of Drug Sciences, Medicinal Chemistry Section, University of Catania, Viale A. Doria 6, I-95125 Catania, Italy

7. Unit of Endocrinology, Department Biomedical, Metabolic, and Neural Sciences, University of Modena and Reggio Emilia, via G. Campi 287, 41125 Modena, Italy

8. Center for Genomic Research, University of Modena and Reggio Emilia, via G. Campi 287, 41125 Modena, Italy

9. Department of Pharmacy, Medicinal Chemistry Section, School of Medical and Pharmaceutical Sciences, University of Genova, Viale Benedetto XV 3, 16132 Genova, Italy

10. Department of Medicinal Chemistry, Maj Institute of Pharmacology, Polish Academy of Sciences, 12, Smętna Street, 31-343, Kraków, Poland

Funder

Ministero dell?Istruzione, dell?Universit? e della Ricerca

Banca d'Italia

Finanziamento annuale individuale delle attivita' base di ricerca

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

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