Discovery of a Novel Muscarinic Receptor PET Radioligand with Rapid Kinetics in the Monkey Brain-Reference-Cited by-同舟云学术

Discovery of a Novel Muscarinic Receptor PET Radioligand with Rapid Kinetics in the Monkey Brain

Published:2017-11-13 Issue:2 Volume:9 Page:224-229
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Malmquist Jonas¹,Varnäs Katarina¹,Svedberg Marie¹,Vallée Frédéric²,Albert Jeffrey S.²,Finnema Sjoerd J.¹,Schou Magnus¹³^ORCID

Affiliation:

1. Department of Clinical Neuroscience, Center for Psychiatry Research, Karolinska Institutet and Stockholm Country Council, SE-171 76 Stockholm, Sweden

2. IntelliSyn Pharma, Montreal H4S 1Z9, Canada

3. PET Science Centre at Karolinska Institutet, Personalised Healthcare and Biomarkers, AstraZeneca R&D, SE-171 76 Stockholm, Sweden

Funder

AstraZeneca

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.7b00340

Reference18 articles.

1. Effect of amphetamine on extrastriatal D2 dopamine receptor binding in the primate brain: A PET study

2. Changes in striatal D2-receptor density following chronic treatment with amphetamine as assessed with pet in nonhuman primates

3. Application of cross-species PET imaging to assess neurotransmitter release in brain

4. Mapping muscarinic receptors in human and baboon brain using [N-11C-methyl]-benztropine

5. In vivo Muscarinic Cholingeric Receptor Imaging in Human Brain with [11C]Scopolamine and Positron Emission Tomography

Cited by 7 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Imaging Cholinergic Receptors in the Brain by Positron Emission Tomography;Journal of Medicinal Chemistry;2023-08-16

2. Update on PET Tracer Development for Muscarinic Acetylcholine Receptors;Pharmaceuticals;2021-06-02

3. Spatial topography of the basal forebrain cholinergic projections: Organization and vulnerability to degeneration;Handbook of Clinical Neurology;2021

4. Enhanced arecoline derivatives as muscarinic acetylcholine receptor M1 ligands for potential application as PET radiotracers;European Journal of Medicinal Chemistry;2020-10

5. First-in-Human Assessment of 11C-LSN3172176, an M1 Muscarinic Acetylcholine Receptor PET Radiotracer;Journal of Nuclear Medicine;2020-08-28