Identification of 5-(1-Methyl-5-(trifluoromethyl)-1H-pyrazol-3-yl)thiophene-2-Carboxamides as Novel and Selective Monoamine Oxidase B Inhibitors Used to Improve Memory and Cognition-Reference-Cited by-同舟云学术

Identification of 5-(1-Methyl-5-(trifluoromethyl)-1H-pyrazol-3-yl)thiophene-2-Carboxamides as Novel and Selective Monoamine Oxidase B Inhibitors Used to Improve Memory and Cognition

Published:2017-09-20 Issue:12 Volume:8 Page:2746-2758
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Kaplan Alan P.¹^ORCID,Keenan Terence¹,Scott Roderick¹,Zhou Xianbo²,Bourchouladze Rusiko¹,McRiner Andrew J.³,Wilson Mark E.¹,Romashko Darlene⁴,Miller Regina⁵,Bletsch Matthew⁶,Anderson Gary¹,Stanley Jennifer¹,Zhang Adia¹,Lee Dong¹,Nikpur John¹

Affiliation:

1. Dart NeuroScience, LLC, 12278 Scripps Summit Drive, San Diego, California 92131, United States

2. SJN Biomed LTD, 398 West Second Ring Road, Kunming 650118, China

3. X-Chem Pharmaceuticals, Inc., 100 Beaver Street, Suite 101, Waltham, Massachusetts 02453, United States

4. Aset Therapeutics, 25 Health Sciences Drive, Stony Brook, New York 11790, United States

5. Bristol-Myers Squibb, 5 Research Parkway, Wallingford, Connecticut 06492, United States

6. The Hain Celestial Group, 1111 Marcus Avenue, New Hyde Park, New York 11042, United States

Funder

Helicon Therapeutics, Inc.

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.7b00282

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