An Improved Process for the N-Alkylation of Indoles Using Chiral N-Protected 2-Methylaziridines-Reference-Cited by-同舟云学术

An Improved Process for the N-Alkylation of Indoles Using Chiral N-Protected 2-Methylaziridines

Published:2002-11-14 Issue:1 Volume:7 Page:22-24
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Giles Paul R.¹,Rogers-Evans Mark¹,Soukup Milan¹,Knight John¹

Affiliation:

1. Vernalis Research Ltd., Oakdene Court, 613 Reading Road, Winnersh, Wokingham RG41 5UA, UK, and F. Hoffmann-La Roche Ltd., CH-4070 Basel, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op020078v

Reference6 articles.

1. Reaktionen mit Aziridinen, 52: Tryptamin‐Verbindungen mit Seitenkettensubstitution aus Indolyllithium und aktivierten Aziridinen

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