A New Avenue toward Androgen Receptor Pan-antagonists: C2 Sterically Hindered Substitution of Hydroxy-propanamides-Reference-Cited by-同舟云学术

A New Avenue toward Androgen Receptor Pan-antagonists: C2 Sterically Hindered Substitution of Hydroxy-propanamides

Published:2014-08-28 Issue:17 Volume:57 Page:7263-7279
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Guerrini Andrea¹,Tesei Anna²,Ferroni Claudia¹,Paganelli Giulia²,Zamagni Alice²,Carloni Silvia²,Di Donato Marzia³,Castoria Gabriella³,Leonetti Carlo⁴,Porru Manuela⁴,De Cesare Michelandrea⁵,Zaffaroni Nadia⁵,Beretta Giovanni Luca⁵,Del Rio Alberto¹,Varchi Greta¹

Affiliation:

1. Institute for the Organic Synthesis and Photoreactivity, Italian National Research Council, Via Gobetti 101, 40129 Bologna, Italy

2. I.R.S.T., Istituto Scientifico Romagnolo per lo Studio e la cura dei Tumori, Via P. Maroncelli, 40, 47014 Meldola, Forlì, Italy

3. Department of Biochemistry, Biophysics and General Pathology, II University of Naples, Via L. De Crecchio, 7, 80138 Naples, Italy

4. Experimental Chemotherapy Laboratory, Regina Elena National Cancer Institute, Via delle Messi d’Oro, 156, 00158 Rome, Italy

5. Fondazione IRCCS Istituto Nazionale dei Tumori Milano, Via Amadeo, 42, 20133 Milano, Italy

Funder

Ministero dell'Istruzione, dell'Università e della Ricerca

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm5005122

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