N1-Fluoroalkyltryptophan Analogues: Synthesis and in vitro Study as Potential Substrates for Indoleamine 2,3-Dioxygenase-Reference-Cited by-同舟云学术

N1-Fluoroalkyltryptophan Analogues: Synthesis and in vitro Study as Potential Substrates for Indoleamine 2,3-Dioxygenase

Published:2015-02-05 Issue:3 Volume:6 Page:260-265
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Henrottin Jean¹,Zervosen Astrid¹,Lemaire Christian¹,Sapunaric Frédéric,Laurent Sophie,Van den Eynde Benoit²,Goldman Serge³⁴,Plenevaux Alain¹,Luxen André¹

Affiliation:

1. Cyclotron Research Center, ‡Department of Chemistry, and §Macromolécules Biologiques, Center for Protein Engineering, Université de Liège, Sart-Tilman, B-4000 Liège, Belgium

2. Ludwig Institute for Cancer Research, Brussels Branch and de Duve Institute, Université Catholique de Louvain, B-1200 Brussels, Belgium

3. PET/Biomedical Cyclotron Unit and Department of Nuclear Medicine, Erasme Hospital, Université Libre de Bruxelles, B-1070 Brussels, Belgium

4. Center for Microscopy and Molecular Imaging, Rue Adrienne Bolland 8, B-6041 Gosselies, Belgium

Funder

Région wallonne

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml500385d

Reference37 articles.