Folate–Vinca Alkaloid Conjugates for Cancer Therapy: A Structure–Activity Relationship-Reference-Cited by-同舟云学术

Folate–Vinca Alkaloid Conjugates for Cancer Therapy: A Structure–Activity Relationship

Published:2014-03-11 Issue:3 Volume:25 Page:560-568
ISSN:1043-1802
Container-title:Bioconjugate Chemistry
language:en
Short-container-title:Bioconjugate Chem.

Author:

Leamon Christopher P.¹,Vlahov Iontcho R.¹,Reddy Joseph A.¹,Vetzel Marilynn¹,Santhapuram Hari Krishna R.¹,You Fei¹,Bloomfield Alicia¹,Dorton Ryan¹,Nelson Melissa¹,Kleindl Paul¹,Vaughn Jeremy F.¹,Westrick Elaine¹

Affiliation:

1. Endocyte, Inc., 300 Kent Avenue, West Lafayette, Indiana 47906, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Pharmaceutical Science,Pharmacology,Biomedical Engineering,Bioengineering,Biotechnology

Link

https://pubs.acs.org/doi/pdf/10.1021/bc400441s

Reference20 articles.

1. Comparative preclinical activity of the folate-targetedVinca alkaloid conjugates EC140 and EC145

2. Preclinical Evaluation of EC145, a Folate-VincaAlkaloid Conjugate

3. Design and regioselective synthesis of a new generation of targeted chemotherapeutics. Part 1: EC145, a folic acid conjugate of desacetylvinblastine monohydrazide

4. Folate receptor expression in carcinomas and normal tissues determined by a quantitative radioligand binding assay

5. Differential regulation of folate receptor isoforms in normal and malignant tissues in vivo and in established cell lines. Physiologic and clinical implications

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