Discovery of AZD3199, An Inhaled Ultralong Acting β2 Receptor Agonist with Rapid Onset of Action-Reference-Cited by-同舟云学术

Discovery of AZD3199, An Inhaled Ultralong Acting β2 Receptor Agonist with Rapid Onset of Action

Published:2014-02-11 Issue:4 Volume:5 Page:416-421
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Stocks Michael J.¹,Alcaraz Lilian¹,Bailey Andrew¹,Bonnert Roger¹,Cadogan Elaine¹,Christie Jadeen¹,Dixon John¹,Connolly Stephen¹,Cook Anthony¹,Fisher Adrian¹,Flaherty Alice¹,Humphries Alexander¹,Ingall Anthony¹,Jordan Stephen¹,Lawson Mandy¹,Mullen Alex¹,Nicholls David¹,Paine Stuart¹,Pairaudeau Garry¹,Young Alan¹

Affiliation:

1. Department of Medicinal Chemistry, ‡Department of Bioscience, and §Department of Physical and Metabolic Sciences, AstraZeneca R&D Charnwood, Bakewell Road, Loughborough, Leicestershire LE11 5RH, U.K.

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml4005232

Reference28 articles.

1. Long-Acting Beta-Agonists and their Association with Inhaled Corticosteroids in COPD

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5. Discovery of olodaterol, a novel inhaled β2-adrenoceptor agonist with a 24h bronchodilatory efficacy

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