Histaprodifens: Synthesis, Pharmacological in Vitro Evaluation, and Molecular Modeling of a New Class of Highly Active and Selective Histamine H1-Receptor Agonists-Reference-Cited by-同舟云学术

Histaprodifens: Synthesis, Pharmacological in Vitro Evaluation, and Molecular Modeling of a New Class of Highly Active and Selective Histamine H1-Receptor Agonists

Published:2000-03-01 Issue:6 Volume:43 Page:1071-1084
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Elz Sigurd¹,Kramer Kai¹,Pertz Heinz H.¹,Detert Heiner¹,ter Laak Anton M.¹,Kühne Ronald¹,Schunack Walter¹

Affiliation:

1. Institut für Pharmazie, Freie Universität Berlin, Königin-Luise-Strasse 2+4, D-14195 Berlin (Dahlem), Germany, Institut für Organische Chemie, Johannes Gutenberg-Universität, J.-J. Becherweg 18-20, D-55099 Mainz, Germany, and Forschungsinstitut für Molekulare Pharmakologie, Alfred-Kowalke-Strasse 4, D-10315 Berlin, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm991056a

Reference63 articles.

1. Is histamine an anticonvulsive inhibitory transmitter?

2. Histamine levels and clonic convulsions of electrically-induced seizure in mice: the effects of ?-fluoromethylhistidine and metoprine

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