Conformations of Trypsin-Bound Amidine Inhibitors of Blood Coagulant Factor Xa by Double REDOR NMR and MD Simulations-Reference-Cited by-同舟云学术

Conformations of Trypsin-Bound Amidine Inhibitors of Blood Coagulant Factor Xa by Double REDOR NMR and MD Simulations

Published:1999-09-01 Issue:19 Volume:42 Page:3910-3918
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

McDowell Lynda M.¹,McCarrick Margaret A.¹,Studelska Daniel R.¹,Guilford William J.¹,Arnaiz Damian¹,Dallas Jerry L.¹,Light David R.¹,Whitlow Marc¹,Schaefer Jacob¹

Affiliation:

1. Department of Chemistry, Washington University, St. Louis, Missouri 63130, and Berlex Biosciences, 15049 San Pablo Avenue, Richmond, California 94804

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9900669

Reference27 articles.

1. Evidence That Macrophages in Atherosclerotic Lesions Contain Angiotensin II

2. Discovery of N-[2-[5-[Amino(imino)methyl]-2-hydroxyphenoxy]-3,5-difluoro- 6-[3-(4,5-dihydro-1-methyl-1H-imidazol-2-yl)phenoxy]pyridin-4-yl]-N-methylglycine (ZK-807834): A Potent, Selective, and Orally Active Inhibitor of the Blood Coagulation Enzyme Factor Xa

3. Synthetic inhibitors of bovine factor Xa and thrombin comparison of their anticoagulant efficiency

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