Initial Scale-Up and Process Improvements for the Preparation of a Lead Antibacterial Macrolone Compound
Author:
Affiliation:
1. GlaxoSmithKline Research Centre, Zagreb Ltd., Prilaz baruna Filipovića 29, HR-10000 Zagreb, Croatia
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/op100199t
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1. Novel 8a-aza-8a-homoerythromycin—4″-(3-substituted-amino)propionates with broad spectrum antibacterial activity
2. 4″-O-(ω-Quinolylamino-alkylamino)propionyl derivatives of selected macrolides with the activity against the key erythromycin resistant respiratory pathogens
3. 6-Alkylquinolone-3-carboxylic acid tethered to macrolides synthesis and antimicrobial profile
4. Synthesis and biological activity of 4″-O-acyl derivatives of 14- and 15-membered macrolides linked to ω-quinolone-carboxylic unit
5. Development of Pd–Cu catalyzed cross-coupling of terminal acetylenes with sp2-carbon halides
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