Asymmetric Reduction of a 1,5-Benzothiazepine Derivative with Sodium Borohydride−(S)-α-Amino Acids: An Efficient Synthesis of a Key Intermediate of Diltiazem-Reference-Cited by-同舟云学术

Asymmetric Reduction of a 1,5-Benzothiazepine Derivative with Sodium Borohydride−(S)-α-Amino Acids: An Efficient Synthesis of a Key Intermediate of Diltiazem

Published:1996-01-01 Issue:24 Volume:61 Page:8586-8590
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Yamada Shin-ichi¹,Mori Yoshikazu¹,Morimatsu Katsuji¹,Ishizu Yoshinori¹,Ozaki Yasuhiko¹,Yoshioka Ryuzo¹,Nakatani Tadashi¹,Seko Hiroyasu¹

Affiliation:

1. Pharmaceutical Development Research Laboratory, Tanabe Seiyaku Co., Ltd., 16-89, Kashima-3-chome, Yodogawa-ku, Osaka 532, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo960950w

Reference45 articles.

1. Synthesis of 1, 5-Benzothiazepine Derivatives. III

2. (c) Abe, K.; Inoue, H.; Nagao, T.Yakugaku Zasshi1988,108, 716.

3. (a) Inoue, H.; Takeo, S.; Kawazu, M.; Kugita, H.Yakugaku Zasshi1973,93, 729.

4. The practical resolution of (2RS,3RS)-2-hydroxy-3-(4-methoxyphenyl)-3-(2-nitrophenylthio)propionic acid, a key intermediate for diltiazem, with L-lysine.

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