Class II (IIa)-Selective Histone Deacetylase Inhibitors. 1. Synthesis and Biological Evaluation of Novel (Aryloxopropenyl)pyrrolyl Hydroxyamides-Reference-Cited by-同舟云学术

Class II (IIa)-Selective Histone Deacetylase Inhibitors. 1. Synthesis and Biological Evaluation of Novel (Aryloxopropenyl)pyrrolyl Hydroxyamides

Published:2005-04-07 Issue:9 Volume:48 Page:3344-3353
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mai Antonello¹,Massa Silvio¹,Pezzi Riccardo¹,Simeoni Silvia¹,Rotili Dante¹,Nebbioso Angela¹,Scognamiglio Annamaria¹,Altucci Lucia¹,Loidl Peter¹,Brosch Gerald¹

Affiliation:

1. Istituto Pasteur - Fondazione Cenci Bolognetti, Dipartimento di Studi Farmaceutici, Università degli Studi di Roma “La Sapienza”, P.le A. Moro 5, 00185 Roma, Italy, Dipartimento Farmaco Chimico Tecnologico, Università degli Studi di Siena, via A. Moro, 53100 Siena, Italy, Dipartimento di Patologia Generale, Seconda Università degli Studi di Napoli, vico L. De Crecchio 7, 80138 Napoli, Italy, Centro di Oncogenomica AIRC, CEINGE Biotecnologia avanzata, Napoli, and Department of Molecular Biology, Innsbruck...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049002a

Reference87 articles.

1. Nuclear histone acetylases and deacetylases and transcriptional regulation: HATs off to HDACs

2. The language of covalent histone modifications

3. Review: Chromatin Structural Features and Targets That Regulate Transcription

4. Acetylation and chromosomal functions

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