1,2,4-Triazolyl Azabicyclo[3.1.0]hexanes: A New Series of Potent and Selective Dopamine D3 Receptor Antagonists

Author:

Micheli Fabrizio12,Arista Luca3,Bonanomi Giorgio12,Blaney Frank E.45,Braggio Simone12,Capelli Anna Maria42,Checchia Anna12,Damiani Federica6,Di-Fabio Romano12,Fontana Stefano12,Gentile Gabriella12,Griffante Cristiana12,Hamprecht Dieter7,Marchioro Carla42,Mugnaini Manolo12,Piner Jacqui85,Ratti Emiliangelo15,Tedesco Giovanna42,Tarsi Luca12,Terreni Silvia12,Worby Angela45,Ashby Charles R.9,Heidbreder Christian10

Affiliation:

1. Neurosciences Centre of Excellence

2. GlaxoSmithKline Medicines Research Centre, Via Fleming 4, 37135 Verona, Italy

3. Novartis Institute Research, Basel, Switzerland

4. Molecular Discovery Research

5. GlaxoSmithKline Medicines Research Centre, NFSP, Harlow, U.K.

6. European Patent Office, Munich, Germany

7. Boehringer Ingelheim, Milan, Italy

8. Safety Assessment

9. Department of Pharmaceutical Sciences, Saint John’s University, Jamaica, New York 11439

10. Reckitt Benckiser Pharmaceuticals, Richmond, Virginia 23235

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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