Effect of Fluorination on the Pharmacological Profile of 11β Isomers of Fulvestrant in Breast Carcinoma Cells-Reference-Cited by-同舟云学术

Effect of Fluorination on the Pharmacological Profile of 11β Isomers of Fulvestrant in Breast Carcinoma Cells

Published:2009-01-09 Issue:3 Volume:52 Page:883-887
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Agouridas Vangelis¹,Magnier Emmanuel¹,Blazejewski Jean-Claude¹,Laïos Ioanna¹,Cleeren Anny¹,Nonclercq Denis¹,Laurent Guy¹,Leclercq Guy¹

Affiliation:

1. Institut Lavoisier de Versailles, UMR CNRS 8180, Université de Versailles St. Quentin en Yvelines, 45 Avenue des Etats-Unis, 78035 Versailles Cedex, France, Laboratoire J.-C. Heuson de Cancérologie Mammaire, Institut Jules Bordet, Service de Médecine, 1, Université Libre de Bruxelles, 1 Rue Héger-Bordet, B-1000 Brussels, Belgium, and Service d’Histologie et de Cytologie Expérimentale, Faculté de Médecine et de Pharmacie, Université de Mons-Hainaut, 6 Avenue du Champ de Mars, B7000 Mons, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm801154q

Reference28 articles.

1. Structural Insights into the Mode of Action of a Pure Antiestrogen

2. The Human Estrogen Receptor-α Is a Ubiquitinated Protein Whose Stability Is Affected Differentially by Agonists, Antagonists, and Selective Estrogen Receptor Modulators

3. Fulvestrant: an oestrogen receptor antagonist with a novel mechanism of action

4. Pure oestrogen antagonists for the treatment of advanced breast cancer

Cited by 13 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Antagonism of Estrogen Receptor α-Driven Transcription Mediated by AP-1 in Breast Cancer Therapy;Endocrines;2024-03-06

2. Oral SERD, a Novel Endocrine Therapy for Estrogen Receptor-Positive Breast Cancer;Cancers;2024-01-31

3. Design, Synthesis, Biological Evaluation, and Computational Studies of Novel Fluorinated Candidates as PI3K Inhibitors: Targeting Fluorophilic Binding Sites;Journal of Medicinal Chemistry;2021-11-18

4. Hydrolysis of FTOH precursors, a simple method to account for some of the unknown PFAS;Chemosphere;2021-08

5. Polyfluorinated scaffolds in drug discovery;Fluorine in Life Sciences: Pharmaceuticals, Medicinal Diagnostics, and Agrochemicals;2019