Synthesis and Biological Evaluation of Analogues of 7-Chloro-4,5-dihydro-4- oxo-8-(1,2,4-triazol-4-yl)-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylic Acid (TQX-173) as Novel Selective AMPA Receptor Antagonists-Reference-Cited by-同舟云学术

Synthesis and Biological Evaluation of Analogues of 7-Chloro-4,5-dihydro-4- oxo-8-(1,2,4-triazol-4-yl)-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylic Acid (TQX-173) as Novel Selective AMPA Receptor Antagonists

Published:2003-11-26 Issue:1 Volume:47 Page:262-272
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Catarzi Daniela¹,Colotta Vittoria¹,Varano Flavia¹,Calabri Francesca Romana¹,Filacchioni Guido¹,Galli Alessandro¹,Costagli Chiara¹,Carlà Vincenzo¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Polo Scientifico, Universita'degli Studi di Firenze, Via Ugo Schiff, 6, Sesto Fiorentino (FI), Italy, and Dipartimento di Farmacologia Preclinica e Clinica, Universita' degli Studi di Firenze, Viale G. Pieraccini, 6, 50134 Firenze, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030906q

Reference50 articles.

1. Ligands for Glutamate Receptors: Design and Therapeutic Prospects

2. Inhibitors of AMPA and Kainate Receptors

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