Discovery of 1-Amino-5H-pyrido[4,3-b]indol-4-carboxamide Inhibitors of Janus Kinase 2 (JAK2) for the Treatment of Myeloproliferative Disorders-Reference-Cited by-同舟云学术

Discovery of 1-Amino-5H-pyrido[4,3-b]indol-4-carboxamide Inhibitors of Janus Kinase 2 (JAK2) for the Treatment of Myeloproliferative Disorders

Published:2011-09-26 Issue:20 Volume:54 Page:7334-7349
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Lim Jongwon¹,Taoka Brandon¹,Otte Ryan D.¹,Spencer Kerrie¹,Dinsmore Christopher J.¹,Altman Michael D.¹,Chan Grace¹,Rosenstein Craig¹,Sharma Sujata¹,Su Hua-Poo¹,Szewczak Alexander A.¹,Xu Lin¹,Yin Hong¹,Zugay-Murphy Joan¹,Marshall C. Gary¹,Young Jonathan R.¹

Affiliation:

1. Departments of ‡Chemistry, §Oncology, ∥In Vitro Pharmacology, ⊥Chemistry Modeling and Informatics, #Drug Metabolism and Pharmacokinetics, and ∞Structural Chemistry, Merck & Co., Inc., 33 Avenue Louis Pasteur, Boston, Massachusetts 02115, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200909u

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