Structure−Activity Relationships and Binding Mode of Styrylquinolines as Potent Inhibitors of HIV-1 Integrase and Replication of HIV-1 in Cell Culture-Reference-Cited by-同舟云学术

Structure−Activity Relationships and Binding Mode of Styrylquinolines as Potent Inhibitors of HIV-1 Integrase and Replication of HIV-1 in Cell Culture

Published:2000-03-22 Issue:8 Volume:43 Page:1533-1540
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zouhiri Fatima¹,Mouscadet Jean-François¹,Mekouar Khalid¹,Desmaële Didier¹,Savouré Delphine¹,Leh Hervé¹,Subra Frédéric¹,Le Bret Marc¹,Auclair Christian¹,d'Angelo Jean¹

Affiliation:

1. Unité de Chimie Organique, UPRES-A du CNRS 8076, Centre d’Etudes Pharmaceutiques, Université Paris-Sud, 5 rue J.-B. Clément, 92296 Châtenay-Malabry, France; Laboratoire de Physicochimie et de Pharmacologie des Macromolécules Biologiques, UMR du CNRS 8532, Institut Gustave Roussy, PRII, 39 rue Camille Desmoulins, 94805 Villejuif, France; and Laboratoire de Physicochimie et de Pharmacologie des Macromolécules Biologiques, UMR du CNRS 8532, LBPA, Ecole Normale Supérieure de Cachan, 94235 Cachan, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm990467o

Reference31 articles.

1. Quantifying Residual HIV-1 Replication in Patients Receiving Combination Antiretroviral Therapy

2. Persistence of HIV-1 Transcription in Peripheral-Blood Mononuclear Cells in Patients Receiving Potent Antiretroviral Therapy

3. Viral Dynamics in HIV-1 Infection

4. Requirement of active human immunodeficiency virus type 1 integrase enzyme for productive infection of human T-lymphoid cells

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