Synthesis and Serotonergic Activity of 3-[2-(Pyrrolidin-1-yl)ethyl]indoles: Potent Agonists for the h5-HT1D Receptor with High Selectivity over the h5-HT1B Receptor-Reference-Cited by-同舟云学术

Synthesis and Serotonergic Activity of 3-[2-(Pyrrolidin-1-yl)ethyl]indoles: Potent Agonists for the h5-HT1D Receptor with High Selectivity over the h5-HT1B Receptor

Published:1999-02-01 Issue:4 Volume:42 Page:677-690
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sternfeld Francine¹,Guiblin Alexander R.¹,Jelley Richard A.¹,Matassa Victor G.¹,Reeve Austin J.¹,Hunt Peter A.¹,Beer Margaret S.¹,Heald Anne¹,Stanton Josephine A.¹,Sohal Bindi¹,Watt Alan P.¹,Street Leslie J.¹

Affiliation:

1. Chemistry, Biochemistry, and Bioanalytical Departments, Merck, Sharp and Dohme Research Laboratories, Neuroscience Research Centre, Terlings Park, Eastwick Road, Harlow, Essex CM20 2QR, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9805687

Reference32 articles.

1. Classification and nomenclature of somatostatin receptors

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3. 5-HT Receptor Classification and Nomenclature: Towards a Harmonization with the Human Genome

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