Design, Synthesis, and Evaluation of Diarylpyridines and Diarylanilines as Potent Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors-Reference-Cited by-同舟云学术

Design, Synthesis, and Evaluation of Diarylpyridines and Diarylanilines as Potent Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors

Published:2010-11-04 Issue:23 Volume:53 Page:8287-8297
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tian Xingtao¹,Qin Bingjie¹,Wu Zhiyuan¹,Wang Xiaofeng¹,Lu Hong²,Morris-Natschke Susan L.³,Chen Chin Ho⁴,Jiang Shibo²,Lee Kuo-Hsiung³⁵,Xie Lan¹

Affiliation:

1. Beijing Institute of Pharmacology & Toxicology, 27 Tai-Ping Road, Beijing 100850, China

2. Lindsley F. Kimball Research Institute, New York Blood Center, New York, New York 10065, United States

3. Natural Products Research Laboratories, Eshelman School of Pharmacy, University of North Carolina, Chapel Hill, North Carolina 27599-7568, United States

4. Duke University Medical Center, Box 2926, Surgical Oncology Research Facility, Durham, North Carolina 27710, United States

5. Chinese Medicine Research and Development Center, China Medical University and Hospital, Taichung, Taiwan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100738d

Reference23 articles.

1. Mechanism of inhibition of HIV-1 reverse transcriptase by non-nucleoside inhibitors

2. New non-nucleoside reverse transcriptase inhibitors (NNRTIs) in development for the treatment of HIV infections

3. Etravirine: a second-generation NNRTI for treatment-experienced adults with resistant HIV-1 infection

4. Structure and Function of HIV-1 Reverse Transcriptase: Molecular Mechanisms of Polymerization and Inhibition

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