Replacement of Glycine with Dicarbonyl and Related Moieties in Analogues of the C-Terminal Pentapeptide of Cholecystokinin: CCK2 Agonists Displaying a Novel Binding Mode-Reference-Cited by-同舟云学术

Replacement of Glycine with Dicarbonyl and Related Moieties in Analogues of the C-Terminal Pentapeptide of Cholecystokinin: CCK2 Agonists Displaying a Novel Binding Mode

Published:2000-09-19 Issue:20 Volume:43 Page:3614-3623
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bellier Bruno¹,Million Marie-Emmanuelle¹,DaNascimento Sophie¹,Meudal Hervé¹,Kellou Safia¹,Maigret Bernard¹,Garbay Christiane¹

Affiliation:

1. Département de Pharmacochimie Moléculaire et Structurale, U266 INSERM, UMR 8600 CNRS, UFR des Sciences Pharmaceutiques et Biologiques, 4, Avenue de l'Observatoire, 75270 Paris Cedex 06, France, and Laboratoire de Chimie Théorique, S.R.S.M.C. · UMR 7565 CNRS, Université Nancy 1 - Université Henri Poincaré, B.P. 239 - Domaine Scientifique Victor Grimard, 54506 Vandoeuvre-les-nancy Cedex, France.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0000416

Reference36 articles.

1. Evidence for the Neuropeptide Cholecystokinin as an Antagonist of Opiate Analgesia

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