Structure–Activity Relationship Studies of Orally Active Antimalarial 3,5-Substituted 2-Aminopyridines-Reference-Cited by-同舟云学术

Structure–Activity Relationship Studies of Orally Active Antimalarial 3,5-Substituted 2-Aminopyridines

Published:2012-12-14 Issue:24 Volume:55 Page:11022-11030
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

González Cabrera Diego¹,Douelle Frederic¹,Younis Yassir¹,Feng Tzu-Shean¹,Le Manach Claire¹,Nchinda Aloysius T.¹,Street Leslie J.¹,Scheurer Christian²³,Kamber Jolanda²³,White Karen L.⁴,Montagnat Oliver D.⁴,Ryan Eileen⁴,Katneni Kasiram⁴,Zabiulla K. Mohammed⁵,Joseph Jayan T.⁵,Bashyam Sridevi⁵,Waterson David⁶,Witty Michael J.⁶,Charman Susan A.⁴,Wittlin Sergio²³,Chibale Kelly¹⁷

Affiliation:

1. Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa

2. Swiss Tropical and Public Health Institute, Socinstrasse 57, 4002 Basel, Switzerland

3. University of Basel, 4002 Basel, Switzerland

4. Centre for Drug Candidate Optimisation, Monash University (Parkville campus), 381 Royal Parade, Parkville, VIC 3052, Australia

5. Syngene International Ltd., Biocon Park, Plot No. 2 & 3, Bommasandra IV Phase, Jigani Link Road, Bangalore 560099, India

6. Medicines for Malaria Venture, ICC, Route de Pré-Bois 20, P.O. Box 1826, 1215 Geneva, Switzerland

7. Institute of Infectious Disease and Molecular Medicine, University of Cape Town, Rondebosch 7701, South Africa

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm301476b

Reference16 articles.

1. The pathogenic basis of malaria

2. The State of the Art in Anti-Malarial Drug Discovery and Development

3. Novel Approaches to Antimalarial Drug Discovery

4. New medicines to improve control and contribute to the eradication of malaria

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