Synthesis, Biological Activity, and Three-Dimensional Quantitative Structure−Activity Relationship Model for a Series of Benzo[c]quinolizin-3-ones, Nonsteroidal Inhibitors of Human Steroid 5α-Reductase 1-Reference-Cited by-同舟云学术

Synthesis, Biological Activity, and Three-Dimensional Quantitative Structure−Activity Relationship Model for a Series of Benzo[c]quinolizin-3-ones, Nonsteroidal Inhibitors of Human Steroid 5α-Reductase 1

Published:2004-06-08 Issue:14 Volume:47 Page:3546-3560
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Occhiato Ernesto G.¹,Ferrali Alessandro¹,Menchi Gloria¹,Guarna Antonio¹,Danza Giovanna¹,Comerci Alessandra¹,Mancina Rosa¹,Serio Mario¹,Garotta Gianni¹,Cavalli Andrea¹,De Vivo Marco¹,Recanatini Maurizio¹

Affiliation:

1. Department of Organic Chemistry “U. Schiff”, University of Firenze, Via della Lastruccia 13, I-50019 Sesto Fiorentino, Italy, Department of Clinical Physiopathology, Endocrinology Unit, University of Firenze, Viale G. Pieraccini 6, I-50134 Firenze, Italy, Serono International S.P.R.I., 12, Chemin des Aulx, CH-1228 Plan-les Ouates, Geneve, Switzerland, and Department of Pharmaceutical Sciences, University of Bologna, Via Belmeloro 6, I-40126 Bologna, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm031131o

Reference51 articles.

1. Benign Prostatic Hyperplasia: Pathogenesis and Medical Therapy

2. Role of 5α-Reductase Inhibitors in the Treatment of Advanced Prostatic Carcinoma

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