Discovery of a Neuroprotective Chemical, (S)-N-(3-(3,6-Dibromo-9H-carbazol-9-yl)-2-fluoropropyl)-6-methoxypyridin-2-amine [(−)-P7C3-S243], with Improved Druglike Properties-Reference-Cited by-同舟云学术

Discovery of a Neuroprotective Chemical, (S)-N-(3-(3,6-Dibromo-9H-carbazol-9-yl)-2-fluoropropyl)-6-methoxypyridin-2-amine [(−)-P7C3-S243], with Improved Druglike Properties

Published:2014-04-16 Issue:9 Volume:57 Page:3746-3754
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Naidoo Jacinth,De Jesus-Cortes Hector¹,Huntington Paula,Estill Sandi,Morlock Lorraine K.,Starwalt Ruth,Mangano Thomas J.²,Williams Noelle S.,Pieper Andrew A.¹,Ready Joseph M.

Affiliation:

1. Departments of Psychiatry, Neurology, and Veterans Affairs, University of Iowa Carver College of Medicine, 200 Hawkins Avenue, Iowa City, Iowa 52242, United States

2. National Institute of Mental Health Psychoactive Drug Screening Program, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina 27599, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm401919s

Reference28 articles.

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4. bMcKnight, S. L.; Pieper, A. A.; Ready, J. M.; De Brabander, J.Proneurogenic Compounds. U.S. Patent 8,604,074, 2013.

5. cMcKnight, S. L.; Pieper, A. A.; Ready, J. M.; De Brabander, J.Proneurogenic Compounds. U.S. Patent 8,362,277, 2013.

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